Selective estrogen receptor modulator
Selective estrogen receptor modulators (SERMs) are a class of compounds that act on the estrogen receptor. A characteristic that distinguishes these substances from pure receptor agonists and antagon...
Selective estrogen receptor modulator - Wikipedia
Toremifene
Toremifene citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. Licensed in the United States under the brand name Fareston, toremife...
Toremifene - Wikipedia
Phytoserm
PhytoSERM (phyto = plant, SERM = selective estrogen receptor modulator) are botanically derived substances that possess SERM qualities, similar to synthetically manufactured drugs of the same category...
Arzoxifene
Arzoxifene is a selective estrogen receptor modulator. It is a potent estrogen antagonist in mammary and uterine tissue while acting as an estrogen agonist to maintain bone density and lower serum cho...
Arzoxifene - Wikipedia
Afimoxifene
Afimoxifene (4-hydroxytamoxifen) is a selective estrogen receptor modulator which is the active metabolite of tamoxifen. Afimoxifene is a transdermal gel formulation and is being developed by Ascend...
Afimoxifene - Wikipedia
Levormeloxifene
Levormeloxifene is an experimental selective estrogen receptor modulator that was being developed as an alternative to estrogen replacement therapy for the treatment and prevention of postmenopausal b...
Levormeloxifene - Wikipedia
Lasofoxifene
Lasofoxifene (INN) (proposed tradename Fablyn) is a non-steroidal selective estrogen receptor modulator (SERM) which is under development by Pfizer for the prevention and treatment of osteoporosis and...
Lasofoxifene - Wikipedia
Idoxifene
Idoxifene is a non-steroidal estrogen antagonist. It is structurally analogous to tamoxifen.
Idoxifene - Wikipedia
Ormeloxifene
Ormeloxifene (also known as centchroman) is one of the selective estrogen receptor modulators, or SERMs, a class of medication which acts on the estrogen receptor. It is best known as a non-hormonal, ...
Ormeloxifene - Wikipedia
Menerba
Menerba (MF101) is an herbal preparation that acts as a selective estrogen receptor modulator (SERM) which is being studied for its potential to relieve hot flashes associated with menopause. Menerba,...
Clomifene
Clomifene (INN) or clomiphene (USAN) (trademarked as Androxal, Clomid and Omifin, citrate salt Serophene) is a selective estrogen receptor modulator (SERM) that has become the most widely prescribed d...
Clomifene - Wikipedia
Cyclofenil
Cyclofenil (INN, trade names Ondogyne, Sexovid, and others) is a selective estrogen receptor modulator.It was investigated as a possible treatment for scleroderma in the 1980s, but was found to be ine...
Cyclofenil - Wikipedia
Bazedoxifene
Bazedoxifene is a third generation selective estrogen receptor modulator (SERM), developed by Pfizer following the completion of their takeover of Wyeth Pharmaceuticals. In late 2013, Pfizer received ...
Bazedoxifene - Wikipedia
Acolbifene
Acolbifene is a selective estrogen receptor modulator.
Tamoxifen
Tamoxifen is an antagonist of the estrogen receptor in breast tissue via its active metabolite, 4-hydroxytamoxifen. In other tissues such as the endometrium, it behaves as an agonist, and thus may be ...
Tamoxifen - Wikipedia
Raloxifene
Raloxifene (marketed as Evista by Eli Lilly and Company) is an oral selective estrogen receptor modulator (SERM) that has estrogenic actions on bone and anti-estrogenic actions on the uterus and breas...
Raloxifene - Wikipedia
Femarelle (DT56a)
Femarelle (DT56a) is as a selective estrogen receptor modulator (SERM) for the treatment of menopause and bone health. Femarelle contains approximately 322 mg DT56a (a tofu extract) and 108 ...
Trioxifene
Trioxifene (LY-133,314) is a selective estrogen receptor modulator (SERM) with competitive binding activity against estradiol for estrogen receptor {alpha} (ER{alpha}) and antagonistic activity agains...
Trioxifene - Wikipedia